SCHEMBL14686196

SCHEMBL14686196

O=C(CNC(=O)c1ccc(S(=O)(=O)N(Oc2ccc(F)cc2)c2cccc(F)c2)cc1)NCC1CCNCC1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 7/20 0.40
KLKB1 P03952 1/20 0.39
CHRM1 P11229 1/20 0.39
SLC6A9 P48067 1/20 0.38
SLC6A5 Q9Y345 1/20 0.38
ALDH1A1 P00352 1/20 0.38
RAB9A P51151 1/20 0.38
USP5 P45974 1/20 0.38
POLB P06746 1/20 0.37
HTT P42858 1/20 0.37
KDM1A O60341 1/20 0.37
F10 P00742 1/20 0.36
PRSS1 P07477 1/20 0.36
AR P10275 1/20 0.36
ITGB3 P05106 2/20 0.36
ITGA2B P08514 2/20 0.36
PPARA Q07869 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3040716 0.99 CXCR3 (0.39) CXCR3KLKB1CHRM1SLC6A9SLC6A5
SCHEMBL14686207 0.95 CXCR3 (0.41) CXCR3KLKB1CHRM1USP5POLB
SCHEMBL3046480 0.95 CXCR3 (0.38) CXCR3KLKB1CHRM1USP5POLB
Hydrochloric Acid SCHEMBL3053536 0.94 CXCR3 (0.41) CXCR3KLKB1CHRM1USP5POLB
SCHEMBL14686171 0.93 CXCR3 (0.45) CXCR3SLC6A9SLC6A5ALDH1A1RAB9A
Hydrochloric Acid SCHEMBL3043975 0.92 CXCR3 (0.44) CXCR3SLC6A9SLC6A5ALDH1A1RAB9A
SCHEMBL14686174 0.87 CXCR3 (0.46) CXCR3RAB9AUSP5POLBKDM1A
Hydrochloric Acid SCHEMBL3047703 0.86 CXCR3 (0.45) CXCR3RAB9AUSP5POLBKDM1A
SCHEMBL3048107 0.85 KDM4E (0.49)
SCHEMBL14686144 0.85 CXCR3 (0.45) CXCR3USP5POLBKDM1AITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2057116-B1 NEW PHENYLSULFAMOYL BENZAMIDE DERIVATIVES AS BRADYKININ ANTAGONISTS RICHTER GEDEON NYRT (HU) 2013-02-13 EP claimed