SCHEMBL14700075

SCHEMBL14700075

Bc1cccc(NC(=O)Nc2ccc(-c3cc(C(C)=O)n4ncnc(N)c34)cc2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.44
NTRK1 P04629 5/20 0.44
NTRK2 Q16620 5/20 0.44
AURKA O14965 4/20 0.44
LCK P06239 4/20 0.44
FYN P06241 4/20 0.44
LYN P07948 4/20 0.44
FLT3 P36888 4/20 0.44
MAPK9 P45984 4/20 0.44
BLK P51451 4/20 0.44
RPS6KA3 P51812 4/20 0.44
STK3 Q13188 4/20 0.44
ROCK1 Q13464 4/20 0.44
MARK2 Q7KZI7 4/20 0.44
PLK4 O00444 3/20 0.44
ROCK2 O75116 3/20 0.44
ABL1 P00519 3/20 0.44
CSF1R P07333 3/20 0.44
MET P08581 3/20 0.44
KIT P10721 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL59021 0.89 KDR (0.44) KDRNTRK1NTRK2AURKALCK
SCHEMBL58190 0.87 FLT3 (0.42) KDRNTRK1NTRK2AURKALCK
SCHEMBL90885 0.81 ACVRL1 (0.61) FLT3AXLMERTKTYRO3ACVRL1
SCHEMBL60736 0.79 NTRK1 (0.43) KDRNTRK1NTRK2AURKALCK
SCHEMBL57029 0.77 AXL (0.41) KDRNTRK1NTRK2AURKALCK
SCHEMBL59041 0.76 NTRK1 (0.49) KDRNTRK1NTRK2AURKALCK
SCHEMBL60270 0.75 ACVRL1 (0.50) AXLMERTKTYRO3ACVRL1PIK3CD
SCHEMBL59784 0.75 AURKB (0.40) KDRNTRK1NTRK2AURKALCK
SCHEMBL58728 0.75 ACVRL1 (0.44) KDRNTRK1NTRK2AURKALCK
SCHEMBL58313 0.74 KDR (0.59) KDRNTRK1NTRK2AURKALCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957485-B1 SUBSTITUTED 4-AMINO-PYRROLOTRIAZINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER HEALTHCARE LLC (US) 2013-02-13 EP disclosed