SCHEMBL14712563

SCHEMBL14712563

Nc1cccc(Cn2cc(NC(=O)c3n[nH]c4cc(-c5ccc(N)nc5)c(F)cc34)cn2)c1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITK Q08881 11/20 0.66
AURKA O14965 2/20 0.52
DYRK1A Q13627 8/20 0.46
GSK3B P49841 6/20 0.46
CLK2 P49760 1/20 0.46
CLK3 P49761 1/20 0.46
SCD O00767 1/20 0.46
WNT1 P04628 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16163138 0.90 ITK (0.82) ITKAURKADYRK1AGSK3BCLK2
SCHEMBL14712461 0.81 ITK (0.82) ITKAURKADYRK1ACLK2CLK3
SCHEMBL14712554 0.81 ITK (0.68) ITKAURKADYRK1AGSK3BCLK2
SCHEMBL14712581 0.80 ITK (0.66) ITKAURKADYRK1AGSK3BCLK2
SCHEMBL14699075 0.80 ITK (1.00) ITKAURKASCD
SCHEMBL14712458 0.79 ITK (0.54) ITKAURKADYRK1ACLK2CLK3
SCHEMBL14712558 0.79 ITK (0.69) ITKAURKADYRK1AGSK3BCLK2
SCHEMBL14712557 0.79 ITK (0.80) ITKAURKADYRK1ACLK2CLK3
SCHEMBL14712429 0.78 ITK (0.64) ITKAURKADYRK1AWNT1
SCHEMBL14712407 0.78 ITK (0.61) ITKAURKASCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013024011-A1 INDAZOLE COMPOUNDS, COMPOSITIONS AND METHODS OF USE F. HOFFMANN-LA ROCHE AG (CH) 2013-02-21 WO disclosed