SCHEMBL14715427

SCHEMBL14715427

COc1cc2nc(N3CCC(Cc4ccccc4)(OC(=O)NCc4cccnc4)CC3)nc(O)c2cc1OC

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 2/20 0.43
PDGFRA P16234 2/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPK1 P28482 1/20 0.43
PDE10A Q9Y233 1/20 0.43
WHR1 P49842 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
RECQL P46063 1/20 0.42
MAPT P10636 2/20 0.42
USP2 O75604 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
DHODH Q02127 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715376 0.93 WHR1 (0.46) WHR1ADRA1AADRA1B
SCHEMBL14715512 0.92 ADRA1A (0.51) ADRA1AADRA1B
SCHEMBL14715298 0.88 WHR1 (0.44) WHR1ADRA1AADRA1B
SCHEMBL14715442 0.88 WHR1 (0.44) WHR1ADRA1AADRA1B
SCHEMBL2170268 0.88 PDGFRB (0.45) PDGFRBPDGFRAALDH1A1KDM4EMAPK1
SCHEMBL14715403 0.88 WHR1 (0.41) PDGFRBWHR1ADRA1AADRA1B
SCHEMBL14715424 0.87 WHR1 (0.42) WHR1ADRA1AADRA1B
SCHEMBL14715369 0.87 PDE5A (0.44) WHR1
SCHEMBL14715456 0.85 WHR1 (0.39) WHR1ADRA1AADRA1B
SCHEMBL14715262 0.84 ADRA1A (0.56) ALDH1A1KDM4EMAPK1MAPTADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346848-B1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed