SCHEMBL14715653

SCHEMBL14715653

C1CCC1.O=C(O)N[C@H]1CC[C@H](CCN2CCC(Oc3cccc(Cl)c3Cl)CC2)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 14/20 0.55
DRD3 P35462 13/20 0.55
HTR1A P08908 3/20 0.51
DRD4 P21917 3/20 0.51
HTR2A P28223 3/20 0.51
HTR2C P28335 3/20 0.51
ADRA2A P08913 2/20 0.51
DRD1 P21728 2/20 0.51
HTR7 P34969 2/20 0.51
ADRA1A P35348 2/20 0.51
HRH1 P35367 2/20 0.51
HTR2B P41595 2/20 0.51
ABCB11 O95342 1/20 0.51
CHRM2 P08172 1/20 0.51
CHRM1 P11229 1/20 0.51
DRD5 P21918 1/20 0.51
KCNH2 Q12809 1/20 0.51
CHRM4 P08173 1/20 0.50
ADRB1 P08588 1/20 0.50
CHRM5 P08912 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3083298 0.89 DRD2 (0.66) DRD2DRD3HTR1ADRD4HTR2A
SCHEMBL3075424 0.89 DRD2 (0.55) DRD2DRD3HTR1ADRD4HTR2A
SCHEMBL14715658 0.89 DRD2 (0.55) DRD2DRD3HTR1ADRD4HTR2A
SCHEMBL3093404 0.85 DRD3 (0.58) DRD2DRD3HTR2A
Cyclopropane SCHEMBL14715571 0.85 NPC1 (0.48) DRD2DRD3HTR2AHRH1KCNH2
SCHEMBL14715668 0.84 DRD2 (0.53) DRD2DRD3HTR1ADRD4HTR2A
SCHEMBL14715659 0.84 DRD3 (0.72) DRD2DRD3HTR1ADRD4HTR2A
SCHEMBL3079766 0.84 DRD3 (0.72) DRD2DRD3HTR1ADRD4HTR2A
SCHEMBL3087640 0.83 DRD2 (0.71) DRD2DRD3HTR1AHTR2AHTR7
SCHEMBL14715656 0.83 DRD2 (0.53) DRD2DRD3HTR1ADRD4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed