SCHEMBL14715670

SCHEMBL14715670

NC(=O)[C@H]1CC[C@H](CCN2CCC(Oc3ccc(F)cc3Cl)CC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 8/20 0.47
CCR3 P51677 8/20 0.47
KCNH2 Q12809 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3956550 1.00 HRH1 (0.47) HRH1CCR3KCNH2SMN1; SMN2ALDH1A1
SCHEMBL3959462 0.91 HRH1 (0.46) HRH1CCR3KCNH2
SCHEMBL3962626 0.91 HRH1 (0.46) HRH1CCR3KCNH2
SCHEMBL14715697 0.89 HRH1 (0.46) HRH1CCR3KCNH2SMN1; SMN2ALDH1A1
SCHEMBL3963825 0.89 HRH1 (0.46) HRH1CCR3KCNH2SMN1; SMN2ALDH1A1
SCHEMBL3959816 0.87 CACNA1I (0.42) HRH1CCR3KCNH2ALDH1A1
SCHEMBL14715704 0.87 CACNA1I (0.42) HRH1CCR3KCNH2ALDH1A1
SCHEMBL3087685 0.87 DRD3 (0.52)
SCHEMBL3086106 0.87 DRD2 (0.46) HRH1CCR3KCNH2
SCHEMBL3086108 0.87 DRD2 (0.46) HRH1CCR3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed