SCHEMBL14715709

SCHEMBL14715709

O=C(N[C@H]1CC[C@H](CCN2CCC(Oc3c(Cl)cc(F)cc3Cl)CC2)CC1)OC1CCOCC1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 16/20 0.45
HTR2A P28223 15/20 0.45
DRD2 P14416 10/20 0.45
HTR1A P08908 5/20 0.42
DRD4 P21917 3/20 0.42
HTR2C P28335 3/20 0.42
HTR2B P41595 3/20 0.42
DRD1 P21728 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715621 0.90 HTR2A (0.47) DRD3HTR2ADRD2HTR1A
SCHEMBL3083178 0.88 DRD3 (0.55) DRD3HTR2ADRD2
SCHEMBL14715655 0.88 DRD3 (0.45) DRD3HTR2ADRD2HTR1ADRD4
SCHEMBL14715563 0.85 HTR2A (0.47) DRD3HTR2ADRD2HTR1A
SCHEMBL3069391 0.84 DRD3 (0.51) DRD3HTR2ADRD2HTR1ADRD4
SCHEMBL14715617 0.84 DRD3 (0.51) DRD3HTR2ADRD2HTR1ADRD4
SCHEMBL14715634 0.83 DRD3 (0.45) DRD3HTR2ADRD2HTR1ADRD4
SCHEMBL14715668 0.82 DRD2 (0.53) DRD3HTR2ADRD2HTR1ADRD4
SCHEMBL3082089 0.81 DRD3 (0.55) DRD3HTR2ADRD2HTR1A
SCHEMBL3084651 0.81 DRD3 (0.54) DRD3HTR2ADRD2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed