SCHEMBL14717841

SCHEMBL14717841

O=C(CCc1cccc2[nH]ccc12)N[C@H]1CCC[C@@](O)(C#Cc2cccc(Cl)c2)C1.O=C(Cc1ccc2c(c1)OCO2)N[C@H]1CCC[C@@](O)(C#Cc2cccc(Cl)c2)C1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
NPSR1 Q6W5P4 1/20 0.40
SIGMAR1 Q99720 2/20 0.38
MCHR1 Q99705 3/20 0.37
HTT P42858 2/20 0.37
NR1H4 Q96RI1 1/20 0.37
EPHX2 P34913 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HPGD P15428 1/20 0.34
RECQL P46063 1/20 0.34
DRD2 P14416 3/20 0.34
HTR2A P28223 3/20 0.34
DRD3 P35462 3/20 0.34
POLB P06746 2/20 0.34
PARP14 Q460N5 1/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL990820 0.90 HPGD (0.41) MCHR1HTTEPHX2HPGDRECQL
SCHEMBL991456 0.87 SIGMAR1 (0.47) MEN1KMT2ASIGMAR1MCHR1NR1H4
SCHEMBL990289 0.75 EPHX2 (0.53) MEN1KMT2ASIGMAR1EPHX2SMN1; SMN2
SCHEMBL16390663 0.75 EPHX2 (0.53) MEN1KMT2ASIGMAR1EPHX2SMN1; SMN2
SCHEMBL990794 0.73 MDM2 (0.41) EPHX2HPGDTHRB
SCHEMBL990846 0.72 NPC1 (0.46) KMT2ASIGMAR1EPHX2SMN1; SMN2
SCHEMBL990965 0.70 GRM5 (0.44) KMT2AEPHX2HPGDMAPTTHRB
SCHEMBL991006 0.68 GRM5 (0.46) HPGD
SCHEMBL992693 0.68 GRM5 (0.46) HPGD
SCHEMBL990109 0.68 GRM5 (0.42) SIGMAR1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130052644-A1 Predictive Markers Useful in the Treatment of Fragile X Syndrome (FXS) NOVARTIS AG (CH) 2013-02-28 US disclosed