SCHEMBL14720577

SCHEMBL14720577

CCOC(=O)c1ccc(C(Br)=C2CCN(C(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.49
GPR119 Q8TDV5 3/20 0.46
NPSR1 Q6W5P4 2/20 0.45
MAPT P10636 1/20 0.45
ADORA1 P30542 1/20 0.45
RAB9A P51151 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
ALDH1A1 P00352 3/20 0.42
NPC1 O15118 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 2/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
ESR1 P03372 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
ESR2 Q92731 1/20 0.41
CA14 Q9ULX7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14723520 0.87 ATM (0.50) ATMGPR119NPSR1MAPTADORA1
SCHEMBL14338856 0.86 NR1H2 (0.45) GPR119MAPTMEN1KMT2AALDH1A1
SCHEMBL474172 0.84 KMT2A (0.46) GPR119MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL14154600 0.84 GPR119 (0.55) GPR119MAPTMEN1KMT2AALDH1A1
SCHEMBL1602493 0.83 GPR119 (0.50) GPR119
SCHEMBL31705318 0.83 KMT2A (0.47) GPR119MEN1KMT2ALMNAESR2
SCHEMBL1473518 0.82 KDM4E (0.51) GPR119MEN1KMT2AESR1ESR2
SCHEMBL19598956 0.81 GPR119 (0.52) GPR119
SCHEMBL4929719 0.81 KMT2A (0.62) GPR119MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL4033844 0.80 ATM (0.48) ATMGPR119NPSR1MAPTADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed