SCHEMBL14720690

SCHEMBL14720690

COC(=O)c1ccc(C=C2CCN(C(=O)OC(C)(C)C)CC2)c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
ALDH1A1 P00352 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ESR2 Q92731 1/20 0.42
PKM P14618 1/20 0.41
NR1H2 P55055 2/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
F13A1 P00488 1/20 0.40
TGM2 P21980 1/20 0.40
TGM1 P22735 1/20 0.40
TGM3 Q08188 1/20 0.40
MAPT P10636 2/20 0.40
TP53 P04637 1/20 0.40
THRB P10828 1/20 0.40
GRM5 P41594 1/20 0.40
STS P08842 2/20 0.40
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12497730 0.89 NR1H2 (0.42) KMT2AMEN1ALDH1A1L3MBTL1ESR2
SCHEMBL14720680 0.86 SRD5A2 (0.44) KMT2AMEN1ALDH1A1L3MBTL1SRD5A2
SCHEMBL1602307 0.82 OGA (0.46) KMT2AMEN1ALDH1A1PKMNR1H2
SCHEMBL6392515 0.81 GRM5 (0.45) KMT2AMEN1ESR2PKMNR1H2
SCHEMBL29902983 0.80 KMT2A (0.52) KMT2AMEN1ALDH1A1L3MBTL1NR1H2
SCHEMBL10306695 0.80 KMT2A (0.52) KMT2AMEN1ALDH1A1L3MBTL1NR1H2
SCHEMBL7971750 0.80 ESR2 (0.48) KMT2AMEN1ALDH1A1ESR2NR1H2
SCHEMBL20304926 0.79 KMT2A (0.46) KMT2AMEN1ALDH1A1PKMNR1H2
SCHEMBL20333548 0.79 KMT2A (0.46) KMT2AMEN1ALDH1A1PKMNR1H2
SCHEMBL20304927 0.79 KMT2A (0.46) KMT2AMEN1ALDH1A1PKMNR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed