SCHEMBL14720680

SCHEMBL14720680

COC(=O)c1ccc(C=C2CCN(C(=O)O)CC2)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 6/20 0.44
ALDH1A1 P00352 7/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TSHR P16473 1/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 2/20 0.38
GAA P10253 2/20 0.38
HDAC2 Q92769 1/20 0.38
P2RY12 Q9H244 1/20 0.38
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12497256 0.88 ALDH1A1 (0.41) ALDH1A1L3MBTL1TSHRMEN1KMT2A
SCHEMBL14720690 0.86 KMT2A (0.45) SRD5A2ALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL14720705 0.81 ALDH1A1 (0.44) SRD5A2ALDH1A1L3MBTL1TSHRKDM4E
SCHEMBL6194728 0.79 OGA (0.50) SRD5A2ALDH1A1TSHRHDAC2
SCHEMBL12497138 0.78 ALDH1A1 (0.43) ALDH1A1L3MBTL1TSHRMEN1KMT2A
SCHEMBL6392680 0.78 SRD5A1 (0.50) SRD5A2ALDH1A1TSHRKMT2AKDM4E
SCHEMBL12497730 0.76 NR1H2 (0.42) ALDH1A1L3MBTL1MEN1KMT2AKDM4E
SCHEMBL9137801 0.76 POLB (0.43) SRD5A2ALDH1A1MEN1KMT2A
SCHEMBL9139619 0.76 SRD5A2 (0.47) SRD5A2ALDH1A1MEN1KMT2AHSP90AA1
SCHEMBL9138031 0.76 SRD5A2 (0.53) SRD5A2ALDH1A1L3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed