SCHEMBL14722103

SCHEMBL14722103

CN1Cc2cc(NS(=O)(=O)c3c(Cl)cccc3Cl)ccc2NC1=O

nearest known ligand 0.69

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 20/20 0.69
CREBBP Q92793 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16760624 0.93 BRD4 (0.70) BRD4CREBBP
SCHEMBL14723518 0.87 BRD4 (0.78) BRD4CREBBP
SCHEMBL14722707 0.84 BRD4 (0.77) BRD4CREBBP
SCHEMBL14723496 0.82 BRD4 (0.80) BRD4CREBBP
SCHEMBL16760615 0.82 BRD4 (0.73) BRD4CREBBP
SCHEMBL14721529 0.82 BRD4 (0.70) BRD4CREBBP
SCHEMBL14723566 0.82 BRD4 (0.77) BRD4CREBBP
SCHEMBL14721322 0.81 BRD4 (0.79) BRD4CREBBP
SCHEMBL14723089 0.81 BRD4 (0.79) BRD4CREBBP
SCHEMBL14722824 0.80 BRD4 (1.00) BRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027168-A1 NOVEL HETEROCYCLIC COMPOUNDS AS BROMODOMAIN INHIBITORS PFIZER INC. (US) 2013-02-28 WO claimed
US-20170122958-A1 Enzymes Functional Probes UNIVERSITY OF DUNDEE (GB) 2017-05-04 US disclosed
US-20170122958-A1 Enzymes Functional Probes UNIVERSITY OF DUNDEE (GB) 2017-05-04 US disclosed
US-20170122958-A1 Enzymes Functional Probes UNIVERSITY OF DUNDEE (GB) 2017-05-04 US disclosed
EP-3074514-A2 ENZYMES FUNCTIONAL PROBES University Of Dundee (GB) 2016-10-05 EP disclosed
WO-2015079259-A2 ENZYMES FUNCTIONAL PROBES UNIVERSITY OF DUNDEE (GB) 2015-06-04 WO disclosed
WO-2015079259-A2 ENZYMES FUNCTIONAL PROBES UNIVERSITY OF DUNDEE (GB) 2015-06-04 WO disclosed
WO-2013027168-A1 NOVEL HETEROCYCLIC COMPOUNDS AS BROMODOMAIN INHIBITORS PFIZER INC. (US) 2013-02-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170122958-A1 Enzymes Functional Probes BRDT, BRD1, BRD3 BRD4 6/4885CREBBP 254/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.