SCHEMBL14729566

SCHEMBL14729566

COc1cnnc(CI)c1O

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 2/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
ALOX15 P16050 1/20 0.31
ALOX12 P18054 1/20 0.31
MAPK1 P28482 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PKM P14618 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14722201 0.71 PDE10A (0.36) ALDH1A1KDM4ELMNATP53CYP3A4
SCHEMBL29027368 0.62 ALDH1A1 (0.60) ALDH1A1KDM4ELMNATP53CYP3A4
SCHEMBL14123484 0.61 ALDH1A1 (0.38) ALDH1A1KDM4ECYP3A4MAPTMAPK1
SCHEMBL21719324 0.60 ALDH1A1 (0.33) ALDH1A1KDM4E
SCHEMBL6130010 0.59 MAPK1 (0.39) ALDH1A1KDM4ELMNATP53CYP3A4
SCHEMBL14430073 0.58 ERN1 (0.50) ALDH1A1KDM4ELMNAMAPTPKM
SCHEMBL8740138 0.57
SCHEMBL11161976 0.57 ALDH1A1 (0.43) ALDH1A1KDM4ETP53CYP3A4MAPT
SCHEMBL30277307 0.57
SCHEMBL31678550 0.57 ALDH1A1 (0.52) ALDH1A1KDM4ELMNACYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027845-A1 RADIOLABELED COMPOUNDS AND THEIR USE AS RADIOTRACERS FOR QUANTITATIVE IMAGING OF PHOSPHODIESTERASE (PDE10A) IN MAMMALS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed