SCHEMBL14730770

SCHEMBL14730770

C=C(NC1CCNC1)c1ccc2[nH]c3c(c2c1)C(C)(C)CC(C)(C)C3=O

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.37
KDR P35968 1/20 0.36
TLR9 Q9NR96 5/20 0.35
TLR8 Q9NR97 5/20 0.35
TLR7 Q9NYK1 5/20 0.35
BRD4 O60885 2/20 0.34
ATAD2 Q6PL18 2/20 0.34
MAPKAPK2 P49137 5/20 0.33
RAB9A P51151 2/20 0.33
KDM1A O60341 1/20 0.33
FLT3 P36888 1/20 0.33
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14730796 0.90 KDR (0.46) JAK2KDRTLR8TLR7MAPKAPK2
SCHEMBL14730722 0.90 KDR (0.46) JAK2KDRTLR8TLR7MAPKAPK2
SCHEMBL14730766 0.85 RAB9A (0.47) JAK2KDRTLR9TLR8TLR7
SCHEMBL14730725 0.84 RAB9A (0.47) JAK2KDRTLR9TLR8TLR7
SCHEMBL16248395 0.84 RAB9A (0.47) JAK2KDRTLR9TLR8TLR7
SCHEMBL16248387 0.84 RAB9A (0.47) JAK2KDRTLR9TLR8TLR7
SCHEMBL14730798 0.82 RAB9A (0.44) JAK2KDRTLR9TLR8TLR7
SCHEMBL14730764 0.82 RAB9A (0.49) JAK2KDRTLR9TLR8TLR7
SCHEMBL14730703 0.82 KDR (0.44) JAK2KDRTLR8TLR7MAPKAPK2
SCHEMBL14730749 0.82 KDR (0.44) JAK2KDRTLR9TLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026163-A1 HEPATITIS C INHIBITOR COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-02-28 WO disclosed