SCHEMBL14740832

SCHEMBL14740832

Cc1c(-c2ccc3[nH]c(CCN(C)C)cc3c2)[nH]c(=O)c(C(=O)O)c1O

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.33
FFAR1 O14842 4/20 0.32
HRH4 Q9H3N8 2/20 0.32
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
NEK1 Q96PY6 1/20 0.32
HRH3 Q9Y5N1 1/20 0.31
KDR P35968 1/20 0.31
PTGS2 P35354 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
TSHR P16473 1/20 0.31
BRD4 O60885 1/20 0.31
PIN1 Q13526 1/20 0.31
DAO P14920 1/20 0.31
BACE1 P56817 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17597619 0.80 TLR9 (0.35) MTNR1AMTNR1BMEN1KMT2ADAO
Hydrochloric Acid SCHEMBL17598109 0.79 TLR9 (0.35) MTNR1AMTNR1BMEN1KMT2ADAO
SCHEMBL17597683 0.78 KDR (0.38) KDRKDM4EMEN1KMT2ATSHR
SCHEMBL14745422 0.76 PTGS2 (0.44) PTGS2BRD4
SCHEMBL14744888 0.74 GSK3B (0.44) KDR
Trifluoroacetic Acid SCHEMBL17598072 0.74 KDR (0.36) KDRKDM4ETSHR
SCHEMBL14757693 0.73 HDAC3 (0.35) KDM4ETSHRDAO
Hydrochloric Acid SCHEMBL14746173 0.73 HDAC3 (0.34) KDM4ETSHRDAO
SCHEMBL14740831 0.73 MEN1 (0.31) MEN1KMT2A
Hydrochloric Acid SCHEMBL17597764 0.72 MEN1 (0.30) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2750504-A1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC Therapeutics, Inc. (US) 2014-07-09 EP disclosed
WO-2013033258-A1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC THERAPEUTICS, INC. (US) 2013-03-07 WO disclosed