SCHEMBL14744184

SCHEMBL14744184

CC(C)(C)OC(=O)NCCc1ncc(C(F)(F)F)[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.43
ALDH1A1 P00352 1/20 0.43
GFER P55789 1/20 0.43
CACNA1H O95180 1/20 0.42
CACNA1B Q00975 1/20 0.42
CACNA1C Q13936 1/20 0.42
HTT P42858 1/20 0.41
BCHE P06276 1/20 0.40
STK17B O94768 1/20 0.40
STK17A Q9UEE5 1/20 0.40
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 2/20 0.38
PDK2 Q15119 1/20 0.38
NQO2 P16083 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL14744029 0.81 MMP2 (0.53) NPSR1ALDH1A1GFERHTTBCHE
SCHEMBL14738249 0.80 MMP2 (0.54) NPSR1ALDH1A1GFERHTTBCHE
SCHEMBL9573412 0.74 NPSR1 (0.43) NPSR1ALDH1A1GFERCACNA1HCACNA1B
SCHEMBL12647348 0.73 TDP1 (0.47) NPSR1STK17BSTK17AMEN1GAA
SCHEMBL4713820 0.73 NPSR1 (0.47) NPSR1ALDH1A1GFERHTTBCHE
SCHEMBL20630527 0.73 CACNA1H (0.43) NPSR1GFERCACNA1HCACNA1BCACNA1C
SCHEMBL15244410 0.72 CACNA1B (0.48) NPSR1ALDH1A1GFERCACNA1HCACNA1B
SCHEMBL15244428 0.72 TP53 (0.42) BCHENQO2CKS1BSKP1SKP2
SCHEMBL29099180 0.69 NPSR1 (0.49) NPSR1ALDH1A1GFERHTTBCHE
SCHEMBL1302384 0.69 NPSR1 (0.51) NPSR1ALDH1A1GFERHTTBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2763990-A1 PYRROLOPYRAZINE KINASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2014-08-13 EP disclosed
WO-2013030138-A1 PYRROLOPYRAZINE KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2013-03-07 WO disclosed