SCHEMBL14745507

SCHEMBL14745507

CCc1cc(C(=O)OC(=O)C(F)(F)F)c(=O)[nH]c1-c1ccc(N2C[C@H]3CCN[C@H]3C2)cc1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.31
MTOR P42345 1/20 0.31
KCNH2 Q12809 1/20 0.31
WDR5 P61964 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL14745505 0.87 KDM4E (0.33) PIK3CAMTORKCNH2WDR5
SCHEMBL14744863 0.86 HRH3 (0.41) KCNH2WDR5
SCHEMBL16568542 0.86 KCNH2 (0.34) PIK3CAMTORKCNH2WDR5
SCHEMBL16577240 0.86 KCNH2 (0.34) PIK3CAMTORKCNH2WDR5
SCHEMBL14745237 0.84 CACNA1B (0.35) KCNH2
SCHEMBL14745082 0.84 CACNA1B (0.35) KCNH2
SCHEMBL14745545 0.84 PDE3B (0.32)
SCHEMBL17595147 0.83 CACNA1B (0.33)
SCHEMBL17594910 0.83 CACNA1B (0.33)
SCHEMBL14744882 0.82 EZH2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016039936-A2 MONOCYCLIC SUBSTITUTED 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-03-17 WO claimed
EP-2750505-A1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC Therapeutics, Inc. (US) 2014-07-09 EP claimed
WO-2013033240-A1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC THERAPEUTICS, INC. (US) 2013-03-07 WO claimed
EP-2750505-A1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC Therapeutics, Inc. (US) 2014-07-09 EP disclosed
WO-2013033240-A1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC THERAPEUTICS, INC. (US) 2013-03-07 WO disclosed