SCHEMBL17595147

SCHEMBL17595147

CCc1cc(C(=O)OC(=O)C(F)(F)F)c(=O)[nH]c1-c1ccc(N2C[C@H]3CCC[C@@H](N)[C@H]3C2)cc1

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 2/20 0.33
PARP1 P09874 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30
PRKD3 O94806 1/20 0.30
MAP4K4 O95819 1/20 0.30
PIM1 P11309 1/20 0.30
CLK2 P49760 1/20 0.30
MAP4K2 Q12851 1/20 0.30
CAMK2D Q13557 1/20 0.30
DYRK1A Q13627 1/20 0.30
PIM3 Q86V86 1/20 0.30
AURKB Q96GD4 1/20 0.30
PRKD2 Q9BZL6 1/20 0.30
CLK4 Q9HAZ1 1/20 0.30
STK17A Q9UEE5 1/20 0.30
MAP4K5 Q9Y4K4 1/20 0.30
PTPN11 Q06124 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17594910 1.00 CACNA1B (0.33) CACNA1BPARP1PARP2PDE3BPDE3A
SCHEMBL14745082 0.95 CACNA1B (0.35) CACNA1BPARP1PARP2PRKD3MAP4K4
SCHEMBL14745237 0.95 CACNA1B (0.35) CACNA1BPARP1PARP2PRKD3MAP4K4
SCHEMBL17594875 0.89 CACNA1B (0.38) CACNA1BPARP1PARP2PDE3BPDE3A
Trifluoroacetic Acid SCHEMBL14740932 0.88 DPP4 (0.32) CACNA1BPARP1PARP2PTPN11
Trifluoroacetic Acid SCHEMBL14741140 0.88 DPP4 (0.32) CACNA1BPARP1PARP2PTPN11
SCHEMBL16568225 0.86 KCNH2 (0.33) CACNA1BPARP1PARP2PDE3BPDE3A
SCHEMBL16568753 0.86 KCNH2 (0.33) CACNA1BPARP1PARP2PDE3BPDE3A
SCHEMBL14741105 0.86 CACNA1B (0.31) CACNA1B
SCHEMBL14745075 0.85 PARP1 (0.31) PARP1PARP2PDE3BPDE3APRKD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016039936-A2 MONOCYCLIC SUBSTITUTED 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-03-17 WO claimed