SCHEMBL14746451

SCHEMBL14746451

CS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccc(Cl)cc3OC(F)(F)F)c(F)c2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RORC P51449 19/20 1.00
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
BRD4 O60885 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14746742 0.92 RORC (0.85) RORCCYP2C9CYP2C19
SCHEMBL14744420 0.92 RORC (1.00) RORCCYP2C9CYP2C19
SCHEMBL14754223 0.91 RORC (1.00) RORCCYP2C9CYP2C19
SCHEMBL14754292 0.91 RORC (0.83) RORCCYP2C9CYP2C19
SCHEMBL14754218 0.86 RORC (0.75) RORC
SCHEMBL14744232 0.83 RORC (1.00) RORCCYP2C9CYP2C19
SCHEMBL14744539 0.82 RORC (0.84) RORCCYP2C9CYP2C19
SCHEMBL14754205 0.82 RORC (0.72) RORCCYP2C9CYP2C19
SCHEMBL14744257 0.80 RORC (0.83) RORCCYP2C9CYP2C19
SCHEMBL24032696 0.79 RORC (0.84) RORCCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013029338-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-03-07 WO disclosed
WO-2013029338-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-03-07 WO disclosed