SCHEMBL14764988

SCHEMBL14764988

COC(=O)C1COc2ccc(C(=O)N(NC(C)(C)C)C(=O)c3cc(C)cc(C)c3)c(C)c2O1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.34
RAB9A P51151 4/20 0.33
NPC1 O15118 4/20 0.33
L3MBTL1 Q9Y468 3/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HTT P42858 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
USP2 O75604 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14937148 0.91 NPC1 (0.32) ABCB1RAB9ANPC1L3MBTL1HTT
SCHEMBL6123388 0.90 NPC1 (0.35) RAB9ANPC1L3MBTL1SMN1; SMN2MAPT
SCHEMBL16239577 0.85 ABCB1 (0.33) ABCB1RAB9AHTTCYP3A4CYP2C9
SCHEMBL16239937 0.83 ABCB1 (0.32) ABCB1RAB9AHTTCYP3A4CYP2C9
SCHEMBL5705240 0.83 NPC1 (0.39) RAB9ANPC1SMN1; SMN2MAPTHTT
SCHEMBL13003219 0.82 ABCB1 (0.55) ABCB1HTTCYP3A4CYP2C9CYP2C19
SCHEMBL4659137 0.82 ABCB1 (0.55) ABCB1HTTCYP3A4CYP2C9CYP2C19
SCHEMBL16239512 0.79 STAT3 (0.33) RAB9AL3MBTL1SMN1; SMN2MAPTTSHR
SCHEMBL5054534 0.79 F2RL3 (0.39) RAB9ANPC1L3MBTL1SMN1; SMN2MAPT
SCHEMBL9905363 0.74 PLK1 (0.40) RAB9ANPC1SMN1; SMN2MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013036574-A1 MODIFIED FORMS OF PSEUDOMONAS EXOTOXIN A INTREXON CORPORATION (US) 2013-03-14 WO disclosed