SCHEMBL14765083

SCHEMBL14765083

Cc1nc2c(Br)cccc2[nH]c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.40
PDGFRB P09619 1/20 0.39
FGFR1 P11362 1/20 0.39
FGFR3 P22607 1/20 0.39
FEN1 P39748 1/20 0.38
KDM4E B2RXH2 2/20 0.38
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
NSD2 O96028 1/20 0.38
CASP6 P55212 1/20 0.38
PARP1 P09874 3/20 0.37
CHEK1 O14757 2/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPK10 P53779 1/20 0.37
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10285823 0.82 MGAM (0.50) BRD4PARP1ALDH1A1MAPK10
SCHEMBL3237187 0.79 PARP1 (0.53) KDM4EGRIN1GRIN2BPARP1TNKS
SCHEMBL30196961 0.79 MGAM (0.45) BRD4FEN1KDM4EGRIN2DGRIN3B
SCHEMBL2358644 0.79 PARP1 (0.53) BRD4PDGFRBFGFR1PARP1CHEK1
SCHEMBL14765025 0.79 MGAM (0.45) BRD4FEN1KDM4EGRIN2DGRIN3B
SCHEMBL1701339 0.78 PARP1 (0.53) KDM4EPARP1ALDH1A1
SCHEMBL14765107 0.77 ALDH1A1 (0.50) KDM4EGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL10252257 0.77 PARP1 (0.45) BRD4KDM4EPARP1ALDH1A1TNKS
SCHEMBL16053516 0.76 GRIN2D (0.42) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL30868875 0.74 PDK2 (0.41) BRD4NSD2CASP6PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed