SCHEMBL14765222

SCHEMBL14765222

CC(C)(C)OC(=O)ON1CCC(COc2ccc(B3OC(C)(C)C(C)(C)O3)cc2C#N)CC1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.39
USP30 Q70CQ3 1/20 0.38
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38
XDH P47989 5/20 0.36
GPR119 Q8TDV5 1/20 0.35
IKBKE Q14164 1/20 0.34
TBK1 Q9UHD2 1/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
DGAT1 O75907 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14771892 0.88 USP30 (0.48) AAK1USP30GPR119TBK1
SCHEMBL18339778 0.84 USP30 (0.51) AAK1USP30GPR119TBK1PDE4B
SCHEMBL14771879 0.83 XDH (0.40) USP30XDHIKBKETBK1
SCHEMBL18340579 0.82 USP30 (0.45) AAK1USP30PRMT5WDR77GPR119
SCHEMBL14764910 0.82 AAK1 (0.48) AAK1XDHGPR119PDE4APDE4B
SCHEMBL17323930 0.81 USP30 (0.47) AAK1USP30GPR119TBK1PDE4B
SCHEMBL14764058 0.81 XDH (0.41) XDHIKBKETBK1
SCHEMBL16491266 0.79 USP30 (0.41) AAK1USP30PRMT5WDR77GPR119
SCHEMBL14764331 0.79 XDH (0.43) XDHIKBKETBK1
SCHEMBL23810495 0.77 AAK1 (0.46) AAK1PRMT5WDR77DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013034238-A1 BENZONITRILE DERIVATIVES AS KINASE INHIBITORS MERCK PATENT GMBH (DE) 2013-03-14 WO disclosed