SCHEMBL14765267

SCHEMBL14765267

FC(F)(F)c1ccc(-c2cc(Cl)nn3ccnc23)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 5/20 0.45
NR1D1 P20393 1/20 0.41
DYRK1A Q13627 1/20 0.40
DYRK2 Q92630 1/20 0.40
KCNQ3 O43525 2/20 0.38
KCNQ2 O43526 2/20 0.38
S1PR1 P21453 1/20 0.38
S1PR3 Q99500 1/20 0.38
KIF11 P52732 1/20 0.38
TOP1 P11387 2/20 0.37
JAK3 P52333 4/20 0.36
SRC P12931 1/20 0.34
BRAF P15056 1/20 0.34
KDR P35968 1/20 0.34
CCNB2 O95067 1/20 0.34
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
CCNB3 Q8WWL7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10756085 0.81 KDR (0.34) JAK2NR1D1KDR
SCHEMBL530189 0.81 CDK2 (0.40) KDRCCNB2CDK1CCNB1CCNB3
SCHEMBL23992867 0.75 HTR2C (0.35) JAK2NR1D1DYRK1ADYRK2KCNQ3
SCHEMBL23995238 0.75 HTR2C (0.35) JAK2NR1D1DYRK1ADYRK2KCNQ3
SCHEMBL2588629 0.73 DYRK3 (0.45) DYRK1ADYRK2KDRCYP19A1CYP11B1
SCHEMBL1346284 0.73 JAK2 (0.40) JAK2DYRK1AKCNQ3KCNQ2KIF11
SCHEMBL29892546 0.72 JAK2 (0.39) JAK2DYRK1AKCNQ3KCNQ2KIF11
SCHEMBL30224440 0.71 ERN1 (0.40) JAK2
SCHEMBL23993369 0.70 RAF1 (0.35) NR1D1BRAFKDR
SCHEMBL23993376 0.70 RAF1 (0.35) NR1D1BRAFKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013034048-A1 SUBSTITUTED BENZOFURAN COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES MERCK SHARP & DOHME CORP. (US) 2013-03-14 WO disclosed