SCHEMBL14765610

SCHEMBL14765610

CN1CCN(CCN2CCC(=O)NCCCOc3ccc(CI)cc3Nc3nccc(n3)Nc3cccc(c3)C2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BMPR2 Q13873 1/20 0.37
HTR1A P08908 7/20 0.35
HTR1D P28221 6/20 0.35
HTR1B P28222 6/20 0.35
SLC6A4 P31645 5/20 0.35
PLK4 O00444 1/20 0.34
CDK2 P24941 11/20 0.34
FLT3 P36888 11/20 0.34
JAK2 O60674 10/20 0.34
CCNA2 P20248 10/20 0.34
CCNA1 P78396 10/20 0.34
JAK1 P23458 3/20 0.33
TYK2 P29597 2/20 0.33
ROCK2 O75116 1/20 0.33
CCNK O75909 1/20 0.33
STK10 O94804 1/20 0.33
PRKD3 O94806 1/20 0.33
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33
PRKCB P05771 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL463821 0.92 BMPR2 (0.38) BMPR2HTR1AHTR1DHTR1BPLK4
SCHEMBL415037 0.92 BMPR2 (0.38) BMPR2PLK4CDK2FLT3JAK2
SCHEMBL414518 0.82 BMPR2 (0.39) BMPR2CDK2FLT3JAK2CCNA2
SCHEMBL14765621 0.81 CHEK1 (0.41) JAK2JAK1TYK2MAP4K3JAK3
SCHEMBL416119 0.80 ALK (0.40) FLT3JAK2JAK1TYK2JAK3
SCHEMBL10291311 0.78 BMPR2 (0.39) BMPR2CDK2FLT3JAK2CCNA2
SCHEMBL415035 0.78 BMPR2 (0.39) BMPR2CDK2FLT3JAK2CCNA2
SCHEMBL10290794 0.78 CHEK1 (0.37) FLT3JAK2JAK1TYK2MAP4K3
SCHEMBL14765637 0.78 MAP4K1 (0.37) CDK2FLT3JAK2CCNA2CCNA1
SCHEMBL14765623 0.78 CHEK1 (0.35) FLT3JAK2JAK1TYK2MAP4K3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8394955-B2 2,4 (4,6) pyrimidine derivatives JANSSEN PHARMACEUTICA N.V. (BE) 2013-03-12 US disclosed