SCHEMBL14765634

SCHEMBL14765634

CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4ccccn4)c(CI)c3)c2cc1NC(C)=O

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STK3 Q13188 7/20 0.82
STK4 Q13043 14/20 0.72
EGFR P00533 5/20 0.69
ERBB2 P04626 4/20 0.67
STK25 O00506 1/20 0.64
MAP2K7 O14733 1/20 0.64
CHEK1 O14757 1/20 0.64
GAK O14976 1/20 0.64
EPHB6 O15197 1/20 0.64
ABCC4 O15439 1/20 0.64
MAP3K13 O43283 1/20 0.64
NUAK1 O60285 1/20 0.64
STK17B O94768 1/20 0.64
STK10 O94804 1/20 0.64
PRKD3 O94806 1/20 0.64
ABCB11 O95342 1/20 0.64
MAP4K4 O95819 1/20 0.64
CHEK2 O96017 1/20 0.64
ABL1 P00519 1/20 0.64
INSR P06213 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14765613 0.91 STK3 (0.68) STK3STK4EGFRERBB2STK25
SCHEMBL13826188 0.91 STK3 (0.85) STK3STK4EGFRERBB2STK25
SCHEMBL2384641 0.90 STK3 (1.00) STK3STK4EGFRERBB2STK25
SCHEMBL33532011 0.90 STK3 (1.00) STK3STK4EGFRERBB2STK25
SCHEMBL14765643 0.87 STK4 (0.66) STK3STK4EGFRERBB2STK25
SCHEMBL10054548 0.84 STK4 (0.76) STK3STK4EGFRERBB2STK25
SCHEMBL2384343 0.84 STK3 (0.85) STK3STK4EGFRERBB2STK25
SCHEMBL33531997 0.84 STK3 (0.85) STK3STK4EGFRERBB2STK25
SCHEMBL22419770 0.83 STK4 (1.00) STK3STK4EGFRERBB2STK25
SCHEMBL12309393 0.83 STK4 (0.77) STK3STK4EGFRERBB2STK25

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8394959-B2 Maleate salts of (E)-N-{4-[3-chloro-4-(2-pyridinylmethoxy)anilino]-3-cyano-7-ethoxy-6-quinolinyl)-4-(dimethylamino)-2-buteramide and crystalline forms thereof WYETH LLC (US) 2013-03-12 US disclosed