SCHEMBL14767408

SCHEMBL14767408

OCC1CCN(CCOc2ccc(-c3ccc(-c4ccc(O)cc4)cn3)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 4/20 0.54
ESR1 P03372 6/20 0.50
ESR2 Q92731 6/20 0.50
MCHR1 Q99705 4/20 0.47
CHRM1 P11229 2/20 0.47
HTR2A P28223 2/20 0.47
HRH3 Q9Y5N1 2/20 0.47
ACHE P22303 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12440195 0.90 MCHR1 (0.59) LTA4HMCHR1CHRM1HTR2AHRH3
SCHEMBL14767387 0.86 ESR1 (0.63) LTA4HESR1ESR2MCHR1CHRM1
SCHEMBL4692595 0.86 LTA4H (0.69) LTA4HESR1ESR2HRH3ACHE
SCHEMBL12440214 0.79 MCHR1 (0.59) MCHR1CHRM1HTR2AHRH3
SCHEMBL14767389 0.79 ESR1 (0.60) LTA4HESR1ESR2MCHR1CHRM1
SCHEMBL12440210 0.78 MCHR1 (0.57) MCHR1CHRM1HTR2AHRH3
SCHEMBL12440032 0.77 HRH3 (0.70) LTA4HMCHR1CHRM1HTR2AHRH3
SCHEMBL12441194 0.77 MCHR1 (0.56) MCHR1CHRM1HTR2AHRH3
SCHEMBL12441185 0.77 MCHR1 (0.56) MCHR1CHRM1HTR2AHRH3
SCHEMBL12441099 0.76 MCHR1 (0.72) MCHR1CHRM1HTR2AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558578-B1 NOVEL ALKYNE COMPOUNDS HAVING AN MCH ANTAGONISTIC EFFECT AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM PHARMA (DE) 2013-03-13 EP disclosed