SCHEMBL14775628

SCHEMBL14775628

Cc1nn(-c2ccccc2)c2sc(C(=O)NCC(=O)N3CCC(C)CC3)cc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.64
NPC1 O15118 2/20 0.64
RAB9A P51151 2/20 0.64
ALDH1A1 P00352 10/20 0.61
KDM4E B2RXH2 10/20 0.61
HPGD P15428 9/20 0.61
NPSR1 Q6W5P4 5/20 0.61
LMNA P02545 3/20 0.61
TSHR P16473 3/20 0.61
GLA P06280 1/20 0.61
PKM P14618 1/20 0.61
HSD17B10 Q99714 3/20 0.60
SMN1; SMN2 Q16637 3/20 0.57
POLB P06746 3/20 0.57
USP2 O75604 2/20 0.57
CREBBP Q92793 1/20 0.57
MAPT P10636 8/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
SAE1 Q9UBE0 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL852678 0.93 HTT (0.64) HTTNPC1RAB9AALDH1A1KDM4E
SCHEMBL852752 0.89 ALDH1A1 (0.65) HTTNPC1RAB9AALDH1A1KDM4E
SCHEMBL853189 0.88 ALDH1A1 (0.75) HTTNPC1RAB9AALDH1A1KDM4E
SCHEMBL853789 0.84 HTT (0.64) HTTNPC1RAB9AALDH1A1KDM4E
SCHEMBL854227 0.83 KDM4E (0.71) HTTNPC1RAB9AALDH1A1KDM4E
SCHEMBL14775627 0.82 PDE7A (0.63)
SCHEMBL854762 0.80 ALDH1A1 (0.67) HTTNPC1RAB9AALDH1A1KDM4E
SCHEMBL853404 0.80 HTT (0.84) HTTNPC1RAB9AALDH1A1KDM4E
SCHEMBL853620 0.80 ALDH1A1 (0.77) HTTNPC1RAB9AALDH1A1KDM4E
SCHEMBL852703 0.80 KDM4E (0.71) HTTNPC1RAB9AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1775298-B1 THIENOPYRAZOLE DERIVATIVE HAVING PDE7 INHIBITORY ACTIVITY DAIICHI SANKYO CO LTD (JP) 2013-03-20 EP claimed