SCHEMBL14775682

SCHEMBL14775682

O=C(O)C1=CCCc2cc(Sc3cccc(F)c3)ccc21

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 8/20 0.44
KDM6B O15054 1/20 0.37
BCL2 P10415 1/20 0.37
MCL1 Q07820 1/20 0.37
EPHX1 P07099 1/20 0.36
MGLL Q99685 1/20 0.36
SLC6A9 P48067 1/20 0.35
SIRT5 Q9NXA8 2/20 0.34
DHODH Q02127 1/20 0.33
HAO1 Q9UJM8 1/20 0.33
PARP10 Q53GL7 1/20 0.33
PARP11 Q9NR21 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL641724 0.90 KDM4C (0.39) KDM4CKDM6BBCL2MCL1EPHX1
SCHEMBL2513812 0.82 MAOA (0.42) KDM4CEPHX1
SCHEMBL10110763 0.78 BCL2 (0.44) KDM4CBCL2MCL1
SCHEMBL10110768 0.78 HPGD (0.47) KDM4CBCL2MCL1
SCHEMBL17361744 0.77 KDM4C (0.36) KDM4CKDM6BMGLLHAO1PARP10
SCHEMBL644016 0.77 EPHX1 (0.36) KDM4CEPHX1MGLLSLC6A9HAO1
SCHEMBL27856967 0.77 KDM4C (0.37) KDM4CKDM6BEPHX1MGLLSLC6A9
Hydrochloric Acid SCHEMBL30558475 0.76 KDM4C (0.36) KDM4CMGLLHAO1PARP10PARP11
SCHEMBL644307 0.76 KDM4C (0.36) KDM4CMGLLHAO1PARP10PARP11
SCHEMBL642086 0.72 MAOA (0.54) KDM4CPARP10PARP11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379491-B1 Process for synthesis of amino-methyl tetraline derivatives HOFFMANN LA ROCHE (CH) 2013-03-20 EP disclosed