SCHEMBL14775808

SCHEMBL14775808

COc1ccc(C)c2[nH]c(CCCN(C)CC[C@]3(O)C[C@@H]4CCC[C@H]3c3ccccc34)nc12

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 11/20 0.58
CACNA1C Q13936 10/20 0.58
CYP3A4 P08684 10/20 0.58
CYP2D6 P10635 9/20 0.58
CYP2C9 P11712 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14775966 1.00 CACNA1H (0.58) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL2548169 1.00 CACNA1H (0.58) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL2546919 1.00 CACNA1H (0.58) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL13815513 0.94 CACNA1H (0.60) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL2548530 0.94 CACNA1H (0.60) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL2549624 0.94 CACNA1H (0.60) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL2543631 0.88 CACNA1H (0.73) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL14775891 0.88 CACNA1H (0.73) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL2546599 0.88 CACNA1H (0.73) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL14775925 0.88 CACNA1H (0.73) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350021-B1 BRIDGED TETRAHYDRONAPHTHALENE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2013-03-20 EP disclosed