SCHEMBL14775925

SCHEMBL14775925

COc1cccc2[nH]c(CCCN(C)CC[C@@]3(O)C[C@H]4CCC[C@@H]3c3ccccc34)nc12

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 16/20 0.73
CACNA1C Q13936 13/20 0.73
CYP3A4 P08684 5/20 0.73
CYP2D6 P10635 4/20 0.73
CYP2C9 P11712 2/20 0.73
MAPT P10636 3/20 0.38
CACNA1B Q00975 3/20 0.38
MEN1 O00255 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 2/20 0.38
KCNH2 Q12809 2/20 0.37
NPC1 O15118 1/20 0.37
CACNA1G O43497 1/20 0.37
CACNA1F O60840 1/20 0.37
ABCB11 O95342 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CHRM2 P08172 1/20 0.37
ABCB1 P08183 1/20 0.37
HTR1A P08908 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14775891 1.00 CACNA1H (0.73) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL2543631 1.00 CACNA1H (0.73) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL2546599 1.00 CACNA1H (0.73) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL2548530 0.90 CACNA1H (0.60) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL13815513 0.90 CACNA1H (0.60) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL2549624 0.90 CACNA1H (0.60) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL14775966 0.88 CACNA1H (0.58) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL14775808 0.88 CACNA1H (0.58) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL2546919 0.88 CACNA1H (0.58) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9
SCHEMBL2548169 0.88 CACNA1H (0.58) CACNA1HCACNA1CCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350021-B1 BRIDGED TETRAHYDRONAPHTHALENE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2013-03-20 EP disclosed