SCHEMBL14775869

SCHEMBL14775869

CN(C)C(=O)CN(C)C(=O)[CH]Cc1ccc(C(=O)Nc2cc(-c3cccs3)ccc2N)cc1

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 18/20 0.65
HDAC2 Q92769 4/20 0.59
KCNH2 Q12809 2/20 0.59
HDAC3 O15379 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14775870 0.86 HDAC1 (0.67) HDAC1HDAC2KCNH2
SCHEMBL4419019 0.83 HDAC1 (0.69) HDAC1HDAC2HDAC3
SCHEMBL652224 0.83 HDAC1 (0.67) HDAC1HDAC2KCNH2HDAC3
SCHEMBL2685456 0.83 HDAC1 (0.68) HDAC1HDAC2HDAC3
SCHEMBL14775962 0.82 HDAC1 (0.63) HDAC1HDAC2KCNH2HDAC3
SCHEMBL2686999 0.81 HDAC1 (0.69) HDAC1HDAC2HDAC3
SCHEMBL2686762 0.81 HDAC1 (0.60) HDAC1HDAC2KCNH2HDAC3
SCHEMBL3643999 0.81 HDAC1 (0.72) HDAC1HDAC2HDAC3
SCHEMBL653854 0.80 HDAC1 (0.64) HDAC1HDAC2KCNH2HDAC3
SCHEMBL4520362 0.80 HDAC1 (0.71) HDAC1HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1991226-B1 INHIBITORS OF HISTONE DEACETYLASE MERCK SHARP & DOHME (US) 2013-03-20 EP claimed