SCHEMBL14775870

SCHEMBL14775870

CN(C)C(=O)CN(C)C(=O)CCc1ccc(C(=O)Nc2cc(-c3cccs3)ccc2N)cc1

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 19/20 0.67
HDAC2 Q92769 3/20 0.61
KCNH2 Q12809 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14775869 0.86 HDAC1 (0.65) HDAC1HDAC2KCNH2
SCHEMBL652224 0.84 HDAC1 (0.67) HDAC1HDAC2KCNH2
SCHEMBL4578410 0.84 HDAC1 (0.74) HDAC1HDAC2
SCHEMBL4578962 0.84 HDAC1 (0.79) HDAC1HDAC2
SCHEMBL2685460 0.83 HDAC1 (0.76) HDAC1HDAC2
SCHEMBL14775963 0.83 HDAC1 (0.70) HDAC1HDAC2KCNH2
SCHEMBL2686762 0.82 HDAC1 (0.60) HDAC1HDAC2KCNH2
SCHEMBL3643999 0.82 HDAC1 (0.72) HDAC1HDAC2
SCHEMBL14155914 0.82 HDAC1 (0.78) HDAC1HDAC2
SCHEMBL653854 0.82 HDAC1 (0.64) HDAC1HDAC2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1991226-B1 INHIBITORS OF HISTONE DEACETYLASE MERCK SHARP & DOHME (US) 2013-03-20 EP claimed