SCHEMBL14780753

SCHEMBL14780753

CCc1ccc2[nH]c(-c3n[nH]cc3NC(=O)C3CCN(C(=O)OC(C)(C)C)CC3)nc2c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTPN2 P17706 1/20 0.43
PTPN1 P18031 1/20 0.43
PTPN6 P29350 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
CHEK2 O96017 3/20 0.41
PARP1 P09874 4/20 0.40
PARP2 Q9UGN5 4/20 0.40
JAK1 P23458 1/20 0.40
PRMT5 O14744 4/20 0.40
STS P08842 2/20 0.40
ABL1 P00519 1/20 0.40
RIN1 Q13671 1/20 0.40
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1646327 0.89 PDPK1 (0.44) PTPN2PTPN1PTPN6NPC1RAB9A
SCHEMBL13545035 0.82 TBK1 (0.41) JAK1ABL1
SCHEMBL13374040 0.80 PDPK1 (0.47) ABL1
SCHEMBL8305843 0.79 PDPK1 (0.46) JAK1ABL1
SCHEMBL13375123 0.78 PDPK1 (0.46) NPC1RAB9A
SCHEMBL10240120 0.77 PDPK1 (0.49) JAK1ABL1
SCHEMBL1646953 0.76 TBK1 (0.42)
SCHEMBL12305619 0.76 PDPK1 (0.49) JAK1ABL1
SCHEMBL13374042 0.76 PDPK1 (0.48) NPC1RAB9A
SCHEMBL13373906 0.76 ABL1 (0.49) JAK1ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8399442-B2 Pharmaceutical compounds ASTEX THERAPEUTICS LIMITED (GB) 2013-03-19 US disclosed
US-8399442-B2 Pharmaceutical compounds ASTEX THERAPEUTICS LIMITED (GB) 2013-03-19 US disclosed