SCHEMBL14788196

SCHEMBL14788196

[2H]C([2H])([2H])Oc1cc(Br)cc(OC([2H])([2H])[2H])c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
MEN1 O00255 1/20 0.34
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CYP1A1 P04798 3/20 0.33
CYP1B1 Q16678 3/20 0.33
CYP3A4 P08684 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2E1 P05181 2/20 0.33
CYP2C8 P10632 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2A6 P11509 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP4B1 P13584 2/20 0.33
CYP2B6 P20813 2/20 0.33
CYP3A5 P20815 2/20 0.33
CYP2A7 P20853 2/20 0.33
CYP3A7 P24462 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14788171 0.95 ALDH1A1 (0.52) ALDH1A1MEN1HPGDRAB9AKMT2A
1,3,5-Trimethoxybenzene SCHEMBL31747519 0.86 ALDH1A1 (0.56) ALDH1A1MEN1HPGDKMT2ACYP1A1
1,3,5-Trimethoxybenzene SCHEMBL31747507 0.80 ALDH1A1 (0.69) ALDH1A1MEN1HPGDKMT2ACYP1A1
SCHEMBL202288 0.80 ALDH1A1 (0.69) ALDH1A1MEN1HPGDRAB9AKMT2A
1,3,5-Trimethoxybenzene SCHEMBL31747526 0.80 ALDH1A1 (0.69) ALDH1A1MEN1HPGDKMT2ACYP1A1
SCHEMBL3966378 0.78 ALDH1A1 (0.65) ALDH1A1MEN1HPGDRAB9AKMT2A
SCHEMBL2999328 0.78 ALDH1A1 (0.65) ALDH1A1MEN1HPGDRAB9AKMT2A
SCHEMBL13948171 0.77
SCHEMBL29868308 0.77
SCHEMBL30252964 0.75 ALDH1A1 (0.33) ALDH1A1MEN1HPGDRAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130072457-A1 PYRAZOLYL QUINAZOLINE KINASE INHIBITORS ASTEX THERAPEUTICS LIMITED (GB) 2013-03-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130072457-A1 PYRAZOLYL QUINAZOLINE KINASE INHIBITORS MAP3K5, MAP3K1, MAP4K2 ALDH1A1 3640/4885MEN1 1371/4885HPGD 853/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.