SCHEMBL14795157

SCHEMBL14795157

CN(CCc1ccccc1)C(=O)c1ccc(-c2cnc3[nH]cc(C(=O)O)c3n2)s1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 5/20 0.40
HSD17B1 P14061 2/20 0.39
HDAC1 Q13547 3/20 0.39
LTB4R Q15722 3/20 0.38
LTB4R2 Q9NPC1 3/20 0.38
ABCC1 P33527 1/20 0.38
ROCK2 O75116 2/20 0.38
ROCK1 Q13464 2/20 0.38
AKT3 Q9Y243 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14795122 0.92 SYK (0.38) HSD17B2HSD17B1HDAC1AKT3
SCHEMBL15755924 0.91 HSD17B2 (0.50) HSD17B2HSD17B1HDAC1
SCHEMBL14795162 0.89 PTGFR (0.39)
SCHEMBL14795325 0.89 SYK (0.38) HSD17B2
SCHEMBL14795323 0.86 SYK (0.37)
SCHEMBL14795147 0.86 MAP4K1 (0.46) HSD17B2
SCHEMBL14795219 0.85 SYK (0.40)
SCHEMBL14795119 0.83 HSD17B2 (0.45) HSD17B2HSD17B1HDAC1AKT3
SCHEMBL15755864 0.83 HSD17B2 (0.41) HSD17B2HSD17B1HDAC1
SCHEMBL14795227 0.81 KDM4E (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571880-A1 PYRROLO [2, 3 - B]PYRAZINE - 7 - CARBOXAMIDE DERIVATIVES AND THEIR USE AS JAK AND SYK INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2013-03-27 EP disclosed