SCHEMBL14795463

SCHEMBL14795463

CN1CCN(c2ccc3[nH]c(-c4c(N)c5cc(C(=O)N[C@@H]6CN7CCC6CC7)ccc5[nH]c4=O)nc3c2)CC1

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 18/20 0.62
PDGFRB P09619 16/20 0.62
KDR P35968 16/20 0.62
FLT1 P17948 3/20 0.55
LCK P06239 1/20 0.48
CHEK1 O14757 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3741617 0.84 FGFR1 (0.72) FGFR1PDGFRBKDRFLT1LCK
SCHEMBL14795700 0.82 FGFR1 (0.69) FGFR1PDGFRBKDRFLT1LCK
SCHEMBL13041467 0.81 FGFR1 (0.90) FGFR1PDGFRBKDRFLT1
SCHEMBL14795909 0.81 PDGFRB (0.61) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL14796151 0.81 PDGFRB (0.61) FGFR1PDGFRBKDRFLT1CHEK1
SCHEMBL14796231 0.80 FGFR1 (0.63) FGFR1PDGFRBKDRFLT1LCK
SCHEMBL14796076 0.80 FGFR1 (0.64) FGFR1PDGFRBKDRFLT1LCK
SCHEMBL14795545 0.79 FGFR1 (0.76) FGFR1PDGFRBKDRFLT1LCK
SCHEMBL3381227 0.78 FGFR1 (0.85) FGFR1PDGFRBKDRFLT1
SCHEMBL15910826 0.78 CHEK1 (0.74) FGFR1PDGFRBKDRFLT1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2762475-A1 Pharmaceutically acceptable salts of quinolinone compounds and their medical use Novartis Vaccines and Diagnostics, Inc. (US) 2014-08-06 EP disclosed
EP-2573079-A2 Benzimidazole quinolinones and uses thereof Novartis Vaccines and Diagnostics, Inc. (US) 2013-03-27 EP disclosed