SCHEMBL14802152

SCHEMBL14802152

C[PH](=O)Oc1cccc2c(=O)c3c(O)cc(N4CCOCC4)cc3oc12

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOA P21397 10/20 0.49
PRKDC P78527 5/20 0.47
ATP1A1 P05023 2/20 0.45
ATP1B1 P05026 2/20 0.45
ATP1A3 P13637 2/20 0.45
ATP1B2 P14415 2/20 0.45
ATP1A2 P50993 2/20 0.45
ATP1B3 P54709 2/20 0.45
FXYD2 P54710 2/20 0.45
ATP1A4 Q13733 2/20 0.45
ACHE P22303 1/20 0.43
MAOB P27338 1/20 0.43
EGFR P00533 1/20 0.39
USP8 P40818 1/20 0.38
TOP2A P11388 1/20 0.38
ACE P12821 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5446244 0.88 MAOA (0.64) MAOAPRKDCATP1A1ATP1B1ATP1A3
SCHEMBL14802155 0.85 MAOA (0.49) MAOAPRKDCATP1A1ATP1B1ATP1A3
SCHEMBL14447677 0.83 PRKDC (0.48) MAOAPRKDCATP1A1ATP1B1ATP1A3
SCHEMBL5446315 0.83 MAOA (0.64) MAOAPRKDCATP1A1ATP1B1ATP1A3
SCHEMBL5446303 0.81 PRKDC (0.53) MAOAPRKDCATP1A1ATP1B1ATP1A3
SCHEMBL14468610 0.78 MAOA (0.43) MAOAPRKDCATP1A1ATP1B1ATP1A3
SCHEMBL5448683 0.77 PRKDC (0.49) MAOAPRKDCATP1A1ATP1B1ATP1A3
SCHEMBL5454434 0.77 MGAM (0.63) MAOAPRKDCACE
SCHEMBL5448690 0.73 PRKDC (0.45) MAOAPRKDCATP1A1ATP1B1ATP1A3
SCHEMBL14802151 0.72 PRKDC (0.46) PRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8404681-B2 Xanthones, thioxanthones and acridinones as DNA-PK inhibitors LUITPOLD PHARMACEUTICALS, INC. (US) 2013-03-26 US disclosed