SCHEMBL14828533

SCHEMBL14828533

Cc1c(C(=O)O)c2cccc(F)c2c(=O)n1C(C)c1c[nH]cn1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
GPR139 Q6DWJ6 2/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
KAT2B Q92831 1/20 0.31
HPD P32754 1/20 0.31
DHODH Q02127 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14828547 0.84 KDM4E (0.34) KMT2AMEN1GPR139KDM4EGAA
SCHEMBL2357893 0.82 MEN1 (0.34) KMT2AMEN1GPR139KDM4EGAA
SCHEMBL2834258 0.81 KDM4E (0.43) KMT2AMEN1GPR139KDM4EGAA
SCHEMBL14828543 0.81 F2RL1 (0.41) KMT2AMEN1KAT2BDHODH
SCHEMBL14828541 0.81 ROCK2 (0.36) KMT2AMEN1GPR139KDM4EGAA
SCHEMBL14828558 0.79 TTR (0.34) KMT2AMEN1GPR139KDM4EGAA
SCHEMBL1364883 0.77 CYP2C9 (0.45)
SCHEMBL2359567 0.75
SCHEMBL2830105 0.75 ATM (0.43) KMT2AMEN1KDM4EGAAKAT2B
SCHEMBL2357787 0.73 F2RL1 (0.39) KAT2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8415373-B2 Isoquinolinone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2013-04-09 US claimed
US-8415373-B2 Isoquinolinone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2013-04-09 US disclosed