SCHEMBL14828545

SCHEMBL14828545

Cc1nc(Cn2c(C)c(C(=O)O)c3cccc(F)c3c2=O)cs1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 1/20 0.50
AKR1B1 P15121 2/20 0.39
SCN9A Q15858 2/20 0.39
GNRHR P30968 1/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
KLKB1 P03952 4/20 0.36
KLK1 P06870 4/20 0.36
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36
MAPT P10636 1/20 0.35
RIPK3 Q9Y572 1/20 0.35
ECE1 P42892 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2306409 0.82 GRIN1 (0.36) AKR1B1MEN1KMT2A
SCHEMBL14828565 0.81 PTGDR2 (0.42) GNRHRMEN1KMT2AALDH1A1MAPT
SCHEMBL2357888 0.80 GRIN1 (0.38) AKR1B1MEN1KMT2AALDH1A1TSHR
SCHEMBL3346327 0.80 MAPT (0.43) FEN1MEN1KMT2AALDH1A1TSHR
SCHEMBL14828544 0.79 MAPT (0.37) FEN1AKR1B1MEN1KMT2ATSHR
SCHEMBL14828532 0.79 GLP1R (0.35) AKR1B1MEN1KMT2ATSHR
SCHEMBL2309555 0.79 FEN1 (0.48) FEN1SCN9AALDH1A1MAPT
SCHEMBL14828568 0.79 CYP1B1 (0.39) FEN1AKR1B1SCN9AGNRHRTSHR
SCHEMBL2313634 0.79 GNRHR (0.37) FEN1AKR1B1SCN9AGNRHRMEN1
SCHEMBL14828515 0.79 FEN1 (0.36) FEN1AKR1B1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8415373-B2 Isoquinolinone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2013-04-09 US claimed
US-8415373-B2 Isoquinolinone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2013-04-09 US disclosed