SCHEMBL14828565

SCHEMBL14828565

Cc1c(C(=O)O)c2cccc(F)c2c(=O)n1Cc1c(F)cccc1F

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 5/20 0.42
GNRHR P30968 5/20 0.39
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KMT2A Q03164 3/20 0.37
MEN1 O00255 1/20 0.37
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14828557 0.86 LMNA (0.40) PTGDR2MAPTALDH1A1KMT2AMEN1
SCHEMBL2831862 0.85 CNR2 (0.46) MAPTKDM4EALDH1A1KMT2AMEN1
SCHEMBL2832433 0.85 LMNA (0.38) MAPTKDM4EALDH1A1KMT2AMEN1
SCHEMBL14828548 0.84 PTGDR2 (0.47) PTGDR2TP53MAPT
SCHEMBL2308886 0.84 MEN1 (0.48) PTGDR2TP53KDM4EKMT2AMEN1
SCHEMBL14828516 0.83 RORC (0.42) PTGDR2MAPTALDH1A1KMT2AMEN1
SCHEMBL3346327 0.83 MAPT (0.43) TP53MAPTKDM4EALDH1A1KMT2A
SCHEMBL14828518 0.83 MEN1 (0.34) PTGDR2TP53KMT2AMEN1ATM
SCHEMBL3379736 0.83 MEN1 (0.34) PTGDR2MAPTKDM4EALDH1A1KMT2A
SCHEMBL2313628 0.83 HTR2A (0.36) GNRHRALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8415373-B2 Isoquinolinone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2013-04-09 US claimed
US-8415373-B2 Isoquinolinone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2013-04-09 US disclosed