SCHEMBL14829623

SCHEMBL14829623

O=C(c1ccc2ncc(N3CCCC3)nc2c1)c1c(F)c(O)cc(F)c1F

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD17B14 Q9BPX1 2/20 0.45
HDAC3 O15379 1/20 0.41
HDAC2 Q92769 1/20 0.41
HCAR2 Q8TDS4 2/20 0.39
HPGD P15428 10/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
PIK3CA P42336 1/20 0.38
HRH3 Q9Y5N1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14829518 0.91 HDAC3 (0.52) HSD17B14HDAC3HDAC2HCAR2LMNA
SCHEMBL14829458 0.91 HPGD (0.46) HDAC3HDAC2HCAR2HPGDLMNA
SCHEMBL14829631 0.89 HSD17B14 (0.47) HSD17B14HDAC3HDAC2HCAR2HPGD
SCHEMBL14829746 0.84 HCAR2 (0.43) HSD17B14HDAC3HDAC2HCAR2HPGD
SCHEMBL14829695 0.83 HSD17B14 (0.46) HSD17B14HDAC3HDAC2HCAR2HPGD
SCHEMBL14829805 0.82 HSD17B14 (0.39) HSD17B14HPGD
SCHEMBL14829847 0.81 HCAR2 (0.42) HSD17B14HDAC3HDAC2HCAR2HPGD
SCHEMBL20246640 0.80 HPGD (0.44) HDAC3HDAC2HCAR2HPGDSMN1; SMN2
SCHEMBL14833212 0.80 CYP3A4 (0.39) LMNA
SCHEMBL14829914 0.80 HDAC3 (0.52) HSD17B14HDAC3HDAC2HCAR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9249111-B2 Substituted quinoxalines as B-RAF kinase inhibitors NEUPHARMA, INC. (US) 2016-02-02 US claimed
US-20140343068-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS NEUPHARMA, INC. 2014-11-20 US claimed
WO-2013049701-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS NEUPHARMA, INC. (US) 2013-04-04 WO claimed
US-20170050938-A1 SUBSTITUTED QUINOXALINES AS B-RAF KINASE INHIBITORS NEUPHARMA, INC. 2017-02-23 US disclosed
US-9249111-B2 Substituted quinoxalines as B-RAF kinase inhibitors NEUPHARMA, INC. (US) 2016-02-02 US disclosed
US-20140343068-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS NEUPHARMA, INC. 2014-11-20 US disclosed
WO-2013049701-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS NEUPHARMA, INC. (US) 2013-04-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140343068-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS BRAF, NRAS, RAF1 HSD17B14 265/4885HDAC3 2274/4885HDAC2 2178/4885
US-20170050938-A1 SUBSTITUTED QUINOXALINES AS B-RAF KINASE INHIBITORS BRAF, RAF1, ARAF HSD17B14 1859/4885HDAC3 1559/4885HDAC2 1666/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.