SCHEMBL14833737

SCHEMBL14833737

COc1cccc(/N=C/c2ccc(C)nc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 2/20 0.51
RECQL P46063 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
MAPT P10636 3/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
PTGS2 P35354 1/20 0.43
CHRM5 P08912 1/20 0.43
ALDH1A1 P00352 4/20 0.43
GAA P10253 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALOX12 P18054 1/20 0.43
HTT P42858 1/20 0.42
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15901041 1.00 CYP1A2 (0.51) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14833738 1.00 CYP1A2 (0.51) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14833678 0.86 CYP1A2 (0.51) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL15902151 0.86 CYP1A2 (0.51) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14833679 0.86 CYP1A2 (0.51) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14832119 0.85 CYP1A2 (0.50) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14832266 0.85 MEN1 (0.53) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14832267 0.85 MEN1 (0.53) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14832120 0.85 CYP1A2 (0.50) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14833591 0.83 CYP1A2 (0.54) CYP1A2CYP3A4RECQLTDP1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2760831-A1 VIRAL REPLICATION INHIBITORS Katholieke Universiteit Leuven (BE) 2014-08-06 EP disclosed
WO-2013045516-A1 VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2013-04-04 WO disclosed