SCHEMBL15902151

SCHEMBL15902151

COc1cccc(/N=C\c2ccc(OC)nc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 2/20 0.51
RECQL P46063 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
MAPT P10636 4/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
HSD17B10 Q99714 2/20 0.48
ALDH1A1 P00352 3/20 0.46
LMNA P02545 2/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
PTGS2 P35354 1/20 0.43
CHRM5 P08912 1/20 0.43
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43
TUBA4A P68366 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14833679 1.00 CYP1A2 (0.51) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14833678 1.00 CYP1A2 (0.51) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14832030 0.91 CYP1A2 (0.48) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14832031 0.91 CYP1A2 (0.48) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14832499 0.89 CYP1A2 (0.46) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14832500 0.89 CYP1A2 (0.46) CYP1A2CYP3A4RECQLTDP1HDAC6
SCHEMBL14833781 0.87 TUBB4A (0.46) MAPTALDH1A1LMNAPTGS2TUBB4A
SCHEMBL14833782 0.87 TUBB4A (0.46) MAPTALDH1A1LMNAPTGS2TUBB4A
SCHEMBL15902472 0.87 TUBB4A (0.46) MAPTALDH1A1LMNAPTGS2TUBB4A
SCHEMBL15901041 0.86 CYP1A2 (0.51) CYP1A2CYP3A4RECQLTDP1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12012411-B2 Viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2024-06-18 US disclosed
US-11566025-B2 Viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2023-01-31 US disclosed
US-20220106321-A1 VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2022-04-07 US disclosed
US-11279704-B2 Viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2022-03-22 US disclosed
EP-2978753-B1 NOVEL VIRAL REPLICATION INHIBITORS UNIV LEUVEN KATH (BE) 2020-08-12 EP disclosed
US-20200223845-A1 NOVEL VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2020-07-16 US disclosed
US-10633378-B2 Viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2020-04-28 US disclosed
EP-3617192-A1 VIRAL REPLICATION INHIBITORS Katholieke Universiteit Leuven K.U. Leuven R&D (BE) 2020-03-04 EP disclosed
US-10550123-B2 Viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2020-02-04 US disclosed
US-20190337954-A1 VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2019-11-07 US disclosed
EP-2760831-B1 VIRAL REPLICATION INHIBITORS UNIV LEUVEN KATH (BE) 2019-08-07 EP disclosed
US-20160297810-A1 NOVEL VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2016-10-13 US disclosed
US-20140213586-A1 VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2014-07-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11566025-B2 Viral replication inhibitors EIF2AK2, MAVS, ZC3HAV1 CYP1A2 4117/4885CYP3A4 3288/4885RECQL 45/4885
US-20140213586-A1 VIRAL REPLICATION INHIBITORS EIF2AK2, MAVS, ZC3HAV1 CYP1A2 4117/4885CYP3A4 3288/4885RECQL 45/4885
US-20160297810-A1 NOVEL VIRAL REPLICATION INHIBITORS EIF2AK2, MAVS, IRF3 CYP1A2 4298/4885CYP3A4 3464/4885RECQL 65/4885
US-11279704-B2 Viral replication inhibitors EIF2AK2, MAVS, ZC3HAV1 CYP1A2 4117/4885CYP3A4 3288/4885RECQL 45/4885
US-20190337954-A1 VIRAL REPLICATION INHIBITORS EIF2AK2, MAVS, ZC3HAV1 CYP1A2 4117/4885CYP3A4 3288/4885RECQL 45/4885
US-10633378-B2 Viral replication inhibitors EIF2AK2, MAVS, ZC3HAV1 CYP1A2 4117/4885CYP3A4 3288/4885RECQL 45/4885
US-10550123-B2 Viral replication inhibitors EIF2AK2, MAVS, ZC3HAV1 CYP1A2 4117/4885CYP3A4 3288/4885RECQL 45/4885
US-20220106321-A1 VIRAL REPLICATION INHIBITORS EIF2AK2, MAVS, ZC3HAV1 CYP1A2 4117/4885CYP3A4 3288/4885RECQL 45/4885
US-20200223845-A1 NOVEL VIRAL REPLICATION INHIBITORS EIF2AK2, MAVS, IRF3 CYP1A2 4298/4885CYP3A4 3464/4885RECQL 65/4885
US-12012411-B2 Viral replication inhibitors EIF2AK2, MAVS, ZC3HAV1 CYP1A2 4117/4885CYP3A4 3288/4885RECQL 45/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.