SCHEMBL14845845

SCHEMBL14845845

Cc1cccc(S(=O)(=O)NCc2ccnc3[nH]ccc23)c1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.50
TNNI3K Q59H18 4/20 0.49
IKBKB O14920 4/20 0.45
CHUK O15111 4/20 0.45
NEK1 Q96PY6 5/20 0.44
ALDH1A1 P00352 1/20 0.43
ROCK1 Q13464 1/20 0.42
MEN1 O00255 1/20 0.42
BRAF P15056 1/20 0.42
SLC40A1 Q9NP59 1/20 0.40
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
ALKBH2 Q6NS38 1/20 0.40
ALKBH3 Q96Q83 1/20 0.40
FTO Q9C0B1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14620965 0.86 TNNI3K (0.47) TNNI3KIKBKBCHUKNEK1ROCK1
SCHEMBL857853 0.85 NEK1 (0.53) KMT2AIKBKBCHUKNEK1ALDH1A1
SCHEMBL857664 0.85 ROCK1 (0.48) TNNI3KIKBKBCHUKALDH1A1ROCK1
SCHEMBL13116651 0.85 NEK1 (0.52) TNNI3KIKBKBCHUKNEK1ROCK1
SCHEMBL14845848 0.84 KMT2A (0.50) KMT2AALDH1A1ROCK1MEN1SLC40A1
SCHEMBL857944 0.83 GPBAR1 (0.46) KMT2ATNNI3KIKBKBCHUKBRAF
SCHEMBL857237 0.82 L3MBTL1 (0.58) KMT2ATNNI3KALDH1A1MEN1
SCHEMBL14620964 0.82 L3MBTL1 (0.45) KMT2ATNNI3KIKBKBCHUKNEK1
SCHEMBL857108 0.80 IKBKB (0.48) KMT2ATNNI3KIKBKBCHUKNEK1
SCHEMBL858357 0.80 NEK1 (0.46) TNNI3KIKBKBCHUKNEK1ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8415469-B2 Compounds and methods for kinase modulation, and indications therefor PLEXXIKON INC. (US) 2013-04-09 US disclosed