SCHEMBL14846286

SCHEMBL14846286

O=C(O)CCCN1CC(C(=O)NCCCc2ccc(Cl)c(Cl)c2)=C(O)C1=O

nearest known ligand 0.80

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
LIPG Q9Y5X9 20/20 0.80
LIPC P11150 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14829352 0.95 LIPG (0.80) LIPGLIPC
SCHEMBL14846238 0.89 LIPG (0.91) LIPGLIPC
SCHEMBL14846262 0.89 LIPG (1.00) LIPGLIPC
SCHEMBL14846203 0.89 LIPG (0.80) LIPGLIPC
SCHEMBL14846287 0.89 LIPG (0.81) LIPGLIPC
SCHEMBL14846224 0.88 LIPG (1.00) LIPGLIPC
SCHEMBL17751153 0.88 LIPG (0.77) LIPGLIPC
SCHEMBL14846283 0.88 LIPG (0.89) LIPGLIPC
SCHEMBL14846221 0.88 LIPG (0.90) LIPGLIPC
SCHEMBL14846670 0.88 LIPG (0.80) LIPGLIPC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9249096-B2 Pyrrolinone carboxamide compounds useful as endothelial lipase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2016-02-02 US disclosed
EP-2760828-B1 PYRROLINONE CARBOXAMIDE COMPOUNDS USEFUL AS ENDOTHELIAL LIPASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2015-10-21 EP disclosed
WO-2013049096-A1 PYRROLINONE CARBOXAMIDE COMPOUNDS USEFUL AS ENDOTHELIAL LIPASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2013-04-04 WO disclosed