SCHEMBL14846360

SCHEMBL14846360

NC(=S)NNC(=O)COc1ccc2c(c1)CC(=O)N2

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.52
GAA P10253 1/20 0.42
ATM Q13315 1/20 0.42
SMYD3 Q9H7B4 8/20 0.42
ROCK2 O75116 1/20 0.42
MAOA P21397 1/20 0.42
KCNH2 Q12809 1/20 0.41
JAK3 P52333 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
AHR P35869 1/20 0.40
CRBN Q96SW2 1/20 0.39
EIF2AK2 P19525 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14815695 0.85 MAOB (0.53) MAOBSMYD3ROCK2MAOAKCNH2
SCHEMBL14815914 0.74 MAOB (0.52) MAOBGAASMYD3
SCHEMBL31722184 0.74 MAOA (0.56) MAOBROCK2MAOAKCNH2CRBN
SCHEMBL14815951 0.74 MAOA (0.56) MAOBROCK2MAOAKCNH2CRBN
SCHEMBL27691373 0.74 MAOB (0.50) MAOBGAASMYD3AHREIF2AK2
SCHEMBL7404515 0.72 MAOB (0.65) MAOBMAOAKCNH2AHRCRBN
SCHEMBL689457 0.72 MAOB (0.62) MAOBGAAMAOAKCNH2AHR
SCHEMBL8092883 0.72 MAOB (0.47) MAOBSMYD3ROCK2KCNH2
SCHEMBL11600967 0.72 MAOA (0.60) MAOBROCK2MAOAKCNH2CRBN
SCHEMBL31718406 0.72 MAOA (0.60) MAOBROCK2MAOAKCNH2CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2760856-B1 SELECTIVE NR2B ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2016-09-14 EP disclosed
WO-2013049119-A1 SELECTIVE NR2B ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2013-04-04 WO disclosed