SCHEMBL14856419

SCHEMBL14856419

Cc1cc(=O)oc2cc(NC(=O)[C@H](CC(=O)O)NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(=O)O)NC(=O)OCc3ccccc3)C(C)C)ccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 9/20 0.55
CASP7 P55210 6/20 0.55
CASP1 P29466 5/20 0.55
CASP9 P55211 5/20 0.55
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
TDP1 Q9NUW8 1/20 0.48
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
HPGD P15428 3/20 0.47
RAB9A P51151 2/20 0.47
HSD17B10 Q99714 2/20 0.47
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
CASP4 P49662 3/20 0.46
CASP10 Q92851 3/20 0.46
CASP8 Q14790 2/20 0.46
SIRT5 Q9NXA8 1/20 0.45
NPC1 O15118 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5888314 0.90 MEN1 (0.54) CASP3CASP7CASP1CASP9MEN1
SCHEMBL29419657 0.90 SIRT5 (0.54) CASP3MEN1KMT2ATDP1KDM4E
SCHEMBL29742197 0.90 SIRT5 (0.54) CASP3MEN1KMT2ATDP1KDM4E
SCHEMBL15569405 0.90 SIRT5 (0.54) CASP3MEN1KMT2ATDP1KDM4E
SCHEMBL29419659 0.90 SIRT5 (0.54) CASP3MEN1KMT2ATDP1KDM4E
SCHEMBL29445883 0.87 KDM4E (0.53) CASP3MEN1KMT2ATDP1KDM4E
SCHEMBL1552674 0.87 KDM4E (0.53) CASP3MEN1KMT2ATDP1KDM4E
SCHEMBL29791072 0.87 KDM4E (0.50) MEN1KMT2ATDP1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL8357861 0.86 KDM4E (0.49) MEN1KMT2ATDP1KDM4EALDH1A1
SCHEMBL29470083 0.86 KDM4E (0.52) MEN1KMT2ATDP1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130280269-A1 Manipulation of HSP70 and IRE1Alpha Protein Interactions NATIONAL UNIVERSITY OF IRELAND (IE) 2013-10-24 US disclosed
EP-2580232-A1 MANIPULATION OF HSP70 AND IRE1ALPHA PROTEIN INTERACTIONS National University of Ireland, Galway (IE) 2013-04-17 EP disclosed
WO-2011154908-A1 MANIPULATION OF HSP70 AND IRE1ALPHA PROTEIN INTERACTIONS NATIONAL UNIVERSITY OF IRELAND, GALWAY (IE) 2011-12-15 WO disclosed