SCHEMBL14864876

SCHEMBL14864876

CCc1cc([N+](=O)[O-])ccc1N1Cc2ccccc2S1(=O)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 6/20 0.40
FFAR4 Q5NUL3 6/20 0.40
KMT2A Q03164 4/20 0.39
ALDH1A1 P00352 3/20 0.39
POLB P06746 2/20 0.39
MEN1 O00255 3/20 0.39
MAPT P10636 3/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 2/20 0.38
LMNA P02545 2/20 0.38
RAB9A P51151 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CA12 O43570 2/20 0.37
CA9 Q16790 2/20 0.37
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
TAS1R2 Q8TE23 1/20 0.37
CA2 P00918 1/20 0.37
WDR5 P61964 1/20 0.36
CA1 P00915 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8164137 0.80 ALDH1A1 (0.37) FFAR1FFAR4KMT2AALDH1A1POLB
SCHEMBL14864875 0.73 GAA (0.42) ALDH1A1POLBMAPTGAALMNA
SCHEMBL14864870 0.72 GAA (0.44) ALDH1A1MAPTGAALMNAL3MBTL1
SCHEMBL13236920 0.68 GAA (0.63) KMT2AALDH1A1POLBMEN1MAPT
SCHEMBL13241732 0.65 ALDH1A1 (0.63) KMT2AALDH1A1MEN1MAPTKDM4E
SCHEMBL701594 0.65 MAPT (0.57) KMT2AALDH1A1MEN1MAPTKDM4E
SCHEMBL29978606 0.65 MAPT (0.57) KMT2AALDH1A1MEN1MAPTKDM4E
SCHEMBL7566464 0.64 POLB (0.59) KMT2AALDH1A1POLBMEN1MAPT
SCHEMBL14864874 0.64 ALDH1A1 (0.55) KMT2AALDH1A1POLBMEN1MAPT
SCHEMBL3642120 0.64 ALDH1A1 (0.41) KMT2AALDH1A1POLBMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8420830-B2 Macrocyclic factor VIIa inhibitors useful as anticoagulants BRISTOL-MYERS SQUIBB COMPANY (US) 2013-04-16 US disclosed