SCHEMBL14865108

SCHEMBL14865108

COC(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)Nc1ccccc1)C(C)C

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.67
CYP2C9 P11712 6/20 0.59
CYP2C19 P33261 6/20 0.59
CYP3A4 P08684 5/20 0.59
CYP2D6 P10635 2/20 0.59
CYP1A2 P05177 2/20 0.59
ELANE P08246 7/20 0.55
ALDH1A1 P00352 2/20 0.53
MAPK1 P28482 1/20 0.53
HTT P42858 1/20 0.53
CMA1 P23946 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12292462 1.00 KCNH2 (0.67) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL12034446 0.94 KCNH2 (0.74) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL17527191 0.92 KCNH2 (0.64) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL17490823 0.91 KCNH2 (0.70) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL17490819 0.91 KCNH2 (0.70) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL18648212 0.91 KCNH2 (0.70) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL15127355 0.90 KCNH2 (0.60) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL17527125 0.90 ALDH1A1 (0.57) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL18020257 0.89 KCNH2 (0.59) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL17562027 0.89 KCNH2 (0.61) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2628481-B1 Trisubstituted heterocycles as replication inhibitors of hepatitis C virus HCV ABBVIE BAHAMAS LTD (BS) 2016-02-24 EP disclosed
EP-2853531-A2 Antiviral compounds AbbVie Bahamas Ltd. (BS) 2015-04-01 EP disclosed
EP-2628481-A1 Trisubstituted heterocycles as replication inhibitors of hepatitis C virus HCV AbbVie Bahamas Ltd. (BS) 2013-08-21 EP disclosed
EP-2368890-B1 Hepatitis C virus inhibitors ABBVIE BAHAMAS LTD (BS) 2013-04-17 EP disclosed