SCHEMBL14865291

SCHEMBL14865291

Cc1ccc(N(C)c2ccc(CNC(=O)C3(NC(=O)c4cncnc4)CC3)cc2)c(C)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 5/20 0.51
HDAC1 Q13547 3/20 0.39
KDM1A O60341 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HTT P42858 1/20 0.39
CNR1 P21554 1/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
CTSS P25774 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NAMPT P43490 1/20 0.35
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
CXCR4 P61073 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13128621 0.89 BDKRB1 (0.53) BDKRB1HDAC1KDM1ACYP3A4CYP2C9
SCHEMBL2810040 0.89 BDKRB1 (0.58) BDKRB1CYP3A4CYP2C9CYP2C19KDM4E
SCHEMBL2806049 0.83 BDKRB1 (0.62) BDKRB1HDAC1CYP3A4KDM4EALDH1A1
SCHEMBL2805998 0.82 BDKRB1 (0.57) BDKRB1CNR1CTSLCTSBCTSS
SCHEMBL14865428 0.81 BDKRB1 (0.53) BDKRB1HDAC1KDM1ACYP3A4CYP2C9
SCHEMBL2806959 0.81 BDKRB1 (0.59) BDKRB1HDAC1KDM1ACYP3A4CYP2C9
SCHEMBL12239078 0.80 BDKRB1 (0.54) BDKRB1HDAC1KDM1ACYP3A4CYP2C9
SCHEMBL14865456 0.79 BDKRB1 (0.59) BDKRB1HDAC1CYP3A4CYP2C9CYP2C19
SCHEMBL764432 0.78 BDKRB1 (0.61) BDKRB1HDAC1CYP3A4CYP2C9CYP2C19
SCHEMBL185880 0.77 BDKRB1 (0.47) BDKRB1CYP3A4CYP2C9CYP2C19CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed